Method The target compound was synthesized from clarithromycin via hydrolyzation,acetylation,cyclic carbonatation,oxidation,decarbonatation,acylation,cyclic carbamatation and cyclization.
方法以克拉霉素为始原料,经水解、乙酰化、
碳酸酯化、氧化、脱碳酸酯化、酰化、
氨基甲酸酯化和
等反应
成目标化
物。